Macitentan D4
| Product Name | Macitentan D4 |
|---|---|
| Alternate Names | Macitentan Stable Isotopes, Stable Isotopes of Macitentan |
| CAT No. | CS-O-14938 |
| CAS No. | 1258428-05-5 |
| Category | Stable Isotopes |
| Stock | IN-Stock |
| Mol. Wt. | 592.30 g/mol |
| Mol. For. | C₁₉H₁₆D₄Br₂N₆O₄S |
| Hazardous | This is a Hazardous Compound |
| COA | View Sample COA |
| MSDS | View Sample MSDS |
| Parent API | Macitentan |
| Purity | Not less than 95 % |
| Smileys | O=[S](NC1=NC=NC(OC([2H])([2H])C([2H])([2H])OC2=NC=C(Br)C=N2)=C1C3=CC=C(Br)C=C3)(NCCC)=O |
| Canonical Smiles | CCCNS(=O)(=O)NC1=C(C(=NC=N1)OCCOC2=NC=C(C=N2)Br)C3=CC=C(C=C3)Br |
| InchIKey | JGCMEBMXRHSZKX-LZMSFWOYSA-N |
| Inchl | InChI=1S/C19H20Br2N6O4S/c1-2-7-26-32(28,29)27-17-16(13-3-5-14(20)6-4-13)18(25-12-24-17)30-8-9-31-19-22-10-15(21)11-23-19/h3-6,10-12,26H,2,7-9H2,1H3,(H,24,25,27)/i8D2,9D2 |
| IUPAC | 5-(4-bromophenyl)-6-[2-(5-bromopyrimidin-2-yl)oxy-1,1,2,2-tetradeuterioethoxy]-N-(propylsulfamoyl)pyrimidin-4-amine |
| Controlled | No |
| Shipping | Free for purchase above 1000$ |
| Delivery | In-Stock, products will be dispatched within 24 hours via FedEx for USA, Europe, and other countries. |
| Return | Returns/replacement accepted if you are not satisfied with the quality of the product, (please send us an email with the reason/issues which are facing, within 15 days, after receipt of the product). |
| Ordering | Place your order online or by email sales@clearsynth.com |
Macitentan D4 is a deuterated form of macitentan, a medication used to treat pulmonary arterial hypertension (PAH). PAH is a condition characterized by high blood pressure in the arteries of the lungs, which can lead to heart failure and other complications. Macitentan D4 works by blocking the action of endothelin, a substance that constricts blood vessels and increases blood pressure.
Macitentan D4 is administered orally, typically in tablet form, with or without food. The recommended dosage is usually once daily, but this may vary depending on the severity of the condition and the individual patient's response to treatment. It is important to follow the dosage instructions provided by the healthcare provider and to not exceed the recommended dose.
Macitentan D4 is a stable isotope-labeled compound, meaning that it contains a higher proportion of deuterium than normal, non-labeled macitentan. Deuterium is a stable, non-radioactive isotope of hydrogen that is commonly used in pharmaceuticals as a tracer or a stabilizing agent. Macitentan D4 has the same chemical structure and mechanism of action as macitentan, but its deuterium content may affect its pharmacokinetics, or how the drug is absorbed, distributed, metabolized, and eliminated in the body.
In conclusion, Macitentan D4 is a medication used to treat pulmonary arterial hypertension by blocking the action of endothelin. It is administered orally and has the same chemical structure and mechanism of action as macitentan, but with a higher proportion of deuterium. It is important to follow the dosage instructions provided by the healthcare provider and to not exceed the recommended dose.
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Related Compounds
Macitentan 13C2 D4 | Macitentan ACT-132577-D4 |