Fenoverine D8

Fenoverine D8 is a stable isotope labeled analog of the drug Fenoverine, which is a smooth muscle relaxant used to treat various gastrointestinal disorders. Fenoverine D8 is commonly used in pharmacokinetic studies to track the distribution, metabolism, and excretion of Fenoverine in the body. The chemical formula of Fenoverine D8 is C26H31D8NO3, and it has a molecular weight of 411.63 g/mol. The drug is administered orally and is rapidly absorbed into the bloodstream, with peak plasma concentrations reached within 1-2 hours after ingestion. The half-life of Fenoverine D8 is approximately 3-4 hours, and it is primarily metabolized in the liver and excreted in the urine. Fenoverine D8 works by blocking the calcium channels in smooth muscle cells, which leads to relaxation and decreased muscle tone. This effect helps to relieve the symptoms of various gastrointestinal disorders, including irritable bowel syndrome and functional dyspepsia. While Fenoverine D8 is generally well-tolerated, some individuals may experience side effects such as dizziness, headaches, and gastrointestinal disturbances. It is important to consult with a healthcare provider before taking Fenoverine D8, especially if you have a history of liver or kidney disease or are taking other medications. Overall, Fenoverine D8 is a valuable tool for pharmacological research and can help to improve our understanding of the mechanisms underlying gastrointestinal disorders and their treatment.