(S)-4-Hydroxycarvedilol-D3
| Product Name | (S)-4-Hydroxycarvedilol-D3 |
|---|---|
| Alternate Names | Carvedilol Stable Isotopes, Stable Isotopes of Carvedilol |
| CAT No. | CS-O-46559 |
| CAS No. | 1217853-93-4 (Unlabelled) |
| Category | Stable Isotopes |
| Stock | Enquire |
| Mol. Wt. | 425.50 g/mol |
| Mol. For. | C24H23D3N2O5 |
| Hazardous | This is not a Hazardous Compound |
| COA | View Sample COA |
| MSDS | View Sample MSDS |
| Parent API | Carvedilol |
| Controlled | No |
| Shipping | Free for purchase above 1000$ |
| Delivery | In-Stock, products will be dispatched within 24 hours via FedEx for USA, Europe, and other countries. |
| Return | Returns/replacement accepted if you are not satisfied with the quality of the product, (please send us an email with the reason/issues which are facing, within 15 days, after receipt of the product). |
| Ordering | Place your order online or by email sales@clearsynth.com |
(S)-4-Hydroxycarvedilol-D3 is a deuterium-labeled version of the active metabolite of Carvedilol, a medication used to treat high blood pressure and heart failure. This compound is used in research and clinical settings to study the metabolism and pharmacokinetics of Carvedilol.
The chemical name of (S)-4-Hydroxycarvedilol-D3 is (2S)-1-{[2-(6-methoxy-2,3-dihydro-1H-inden-4-yl)-1-(propan-2-yl)amino]propan-2-yl}oxy-4-(2-hydroxy-3-(propan-2-ylamino)propoxy)indan-1-one-d3. The deuterium-labeled version contains three extra neutrons, which can be used to track the compound in biological systems.
(S)-4-Hydroxycarvedilol-D3 is metabolized in the liver by the cytochrome P450 enzyme system, specifically by the CYP2D6 enzyme. It is converted to glucuronide and sulfate conjugates, which are excreted in the urine. The half-life of (S)-4-Hydroxycarvedilol-D3 is approximately 7-10 hours.
In conclusion, (S)-4-Hydroxycarvedilol-D3 is a useful tool for studying the metabolism and pharmacokinetics of Carvedilol. Its deuterium labeling allows for easy tracking in biological systems, and its metabolism and excretion pathways have been well-characterized.
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Related Compounds
Carvedilol Dimer Impurity D10 | R-Carvedilol-d4 | S-Carvedilol-d4 | Carvedilol D4 | N-Methyl Carvedilol-d3 Hydrochloride Salt | Carvedilol-13C6 | Carvedilol-D5 | Carvedilol-13C3 | O-Desmethyl Carvedilol-d5 |