Baclofen D4 (2,2,4,4-D4)
| Product Name | Baclofen D4 (2,2,4,4-D4) |
|---|---|
| Alternate Names | Baclofen Stable Isotopes, Stable Isotopes of Baclofen |
| CAT No. | CS-T-48544 |
| CAS No. | 70155-52-1 |
| Category | Stable Isotopes |
| Stock | Enquire |
| Mol. Wt. | 217.69 g/mol |
| Mol. For. | C10H8D4ClNO2 |
| Hazardous | This is not a Hazardous Compound |
| COA | View Sample COA |
| MSDS | View Sample MSDS |
| Parent API | Baclofen |
| Smileys | NC([2H])([2H])C(C1=CC=C(Cl)C=C1)C([2H])([2H])C(O)=O |
| Controlled | No |
| Shipping | Free for purchase above 1000$ |
| Delivery | In-Stock, products will be dispatched within 24 hours via FedEx for USA, Europe, and other countries. |
| Return | Returns/replacement accepted if you are not satisfied with the quality of the product, (please send us an email with the reason/issues which are facing, within 15 days, after receipt of the product). |
| Ordering | Place your order online or by email sales@clearsynth.com |
Baclofen D4 (2,2,4,4-D4) is a deuterated form of baclofen, which is a muscle relaxant and antispastic medication. Baclofen D4 is a labeled compound that is commonly used in research studies to study the pharmacokinetics and metabolism of baclofen.
Baclofen D4 is a GABA-B receptor agonist, which means that it binds to and activates GABA-B receptors in the brain and spinal cord. This leads to a decrease in the release of excitatory neurotransmitters, resulting in muscle relaxation and reduction of spasticity. Baclofen D4 has a half-life of approximately 4 hours and is metabolized primarily in the liver.
The deuterium labeling in Baclofen D4 allows for the differentiation between the labeled and unlabeled form of the compound, making it useful in pharmacokinetic studies. It is also used in the development of new drugs that target GABA-B receptors, as it allows researchers to study the effects of the drug on the body in a more precise manner.
In conclusion, Baclofen D4 is a useful compound for researchers studying the pharmacokinetics and metabolism of baclofen, as well as for the development of new drugs that target GABA-B receptors. Its chemical properties make it an effective tool in research studies, providing valuable insights into the mechanisms of action of muscle relaxants and antispastic medications.
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Related Compounds
Baclofen-d5 | Arbaclofen 13C6 | Baclofen 13C6 | Baclofen-d4,15N | Baclofen D4 Hydrochloride | Baclofen hydrochloride 13C6 | S-Baclofen hydrochloride salt 13C6 |